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Mipsagargin (G-202) is a novel thapsigargin-based targeted proagent consisting of a prostate-specific membrane antigen (PSMA)-specific peptide coupled to an analog of the potent sarcoplasmic/endoplasmic reticulum calcium adenosine triphosphatase (SERCA) pump inhibitor Thapsigargin. Mipsagargin is activated by PSMA-mediated cleavage of an inert masking peptide. Mipsagargin has the potential for refractory, advanced or metastatic solid tumours research.
| Molecular Weight | 1409.52 |
| Formula | C66H100N6O27 |
| CAS Number | 1245732-48-2 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
[3] Trine Bundgaard Andersen, et al. Molecules. Thapsigargin--from Thapsia L. to mipsagargin
[4] Nhu Thi Quynh Doan, et al. Steroids. Targeting thapsigargin towards tumors
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