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MIN-101

Cat. No. M8955

All AbMole products are for research use only, cannot be used for human consumption.

MIN-101 Structure
Synonym:

Roluperidone; CYR-101

Size Price Availability Quantity
5mg USD 120 In stock
10mg USD 190 In stock
50mg USD 550 In stock
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Quality Control & Documentation
Biological Activity

MIN-101 (Roluperidone) is a novel compound with affinities for 5-HT2A and sigma-2 receptors with Ki values of 7.53 nM and 8.19 nM, respectively.

Chemical Information
Molecular Weight 366.43
Formula C22H23FN2O2
CAS Number 359625-79-9
Solubility (25°C) DMSO 10 mM
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Davidson M, et al. Am J Psychiatry. Efficacy and Safety of MIN-101: A 12-Week Randomized, Double-Blind, Placebo-Controlled Trial of a New Drug in Development for the Treatment of Negative Symptoms in Schizophrenia.

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Keywords: MIN-101, Roluperidone; CYR-101 supplier, 5-HT Receptor, inhibitors, activators

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