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Mibefradil dihydrochloride (Ro 40-5967 dihydrochloride) is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s of 2.7 μM and 18.6 μM for T-type and L-type currents, respectively).
| Molecular Weight | 568.55 |
| CAS Number | 116666-63-8 |
| Solubility (25°C) | Water ≥ 90 mg/mL |
| Storage | -20°C, sealed |
[3] H A Welker, et al. Clinical pharmacokinetics of mibefradil
[4] B M Massie. Mibefradil: a selective T-type calcium antagonist
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