Free shipping on all orders over $ 500

Mestranol

Cat. No. M3579

All AbMole products are for research use only, cannot be used for human consumption.

Mestranol Structure
Size Price Availability Quantity
25mg USD 35 In stock
50mg USD 50 In stock
100mg USD 70 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Mestranol is the 3-methyl ether of ethinylestradiol. It was the estrogen used in many of the first oral contraceptives. It is a biologically inactive prodrug of ethinylestradiol to which it is demethylated in the liver with a conversion efficiency of 70% (50 ug of mestranol is pharmacokinetically bioequivalent to 35 ug of ethinylestradiol). </

Chemical Information
Molecular Weight 310.43
Formula C21H26O2
CAS Number 72-33-3
Form Solid
Solubility (25°C) DMSO 10 mg/mL
Ethanol 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Martin Perreault, et al. Design of a Mestranol 2-N-Piperazino-Substituted Derivative Showing Potent and Selective in vitro and in vivo Activities in MCF-7 Breast Cancer Models

[2] M Drzdil. Mestranol Spofa

Related Estrogen Receptor Products
Fulvestrant

Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect.

LY500307

LY500307 is a potent, selective estrogen receptor beta agonist with an EC50 of 0.66 nM.

Calcitriol

Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor. *The compound is unstable in solutions, freshly prepared is recommended

Tamoxifen Citrate (ICI 46474)

Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding.

20-Hydroxyecdysone

20-Hydroxyecdysone (Ecdysterone, 20E) is a naturally occurring ecdysteroid hormone which controls the ecdysis (moulting) and metamorphosis of arthropods.

  Catalog
Abmole Inhibitor Catalog




Keywords: Mestranol supplier, Estrogen Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2026 AbMole BioScience. All Rights Reserved.