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MCH TFA (human, mouse, rat) is a potent peptide agonist of MCH-R and exhibits binding IC50 values of 0.3nM and 1.5 nM for MCH1R and MCH2R, respectively. MCH TFA (human, mouse, rat) is a highly sensitive to MCH-2R in a CHO cell line and monitoring mobilization of intracellular calcium with FLIPR, exhibits functional activation EC50 values of 3.9 nM and 0.1nM for human MCH-1R and MCH-2R, respectively.
| Molecular Weight | 2500.86 |
| Formula | C107H161F3N30O28S4 |
| CAS Number | 128315-56-0 (free base) |
| Solubility (25°C) | DMSO 90 mg/mL |
| Storage | -20°C, dry, sealed |
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