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Inolitazone dihydrochloride

Cat. No. M11283

All AbMole products are for research use only, cannot be used for human consumption.

Inolitazone dihydrochloride Structure
Synonym:

Efatutazone dihydrochloride; CS-7017 dihydrochloride; RS5444 dihydrochloride

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Quality Control & Documentation
Biological Activity

Inolitazone dihydrochloride (Efatutazone dihydrochloride) is a PPARγ agonist with high affinity, activity dependent on PPARγ, inhibiting growth, IC50 is 0.8 nM.

Chemical Information
Molecular Weight 575.50662
Formula C27H28Cl2N4O4S
CAS Number 223132-38-5
Solubility (25°C) DMSO ≥ 20 mg/mL
Storage 4°C, dry, sealed
References

[1] Jonathan Wolf Mueller, et al. J Clin Endocrinol Metab. Steroid Sulfation in Adrenal Tumors

[2] Thomas Alec Lightning, et al. Mol Cell Endocrinol. Steroid disulfates - Sulfation double trouble

[3] Zhengxiong Zhou, et al. Sheng Wu Gong Cheng Xue Bao. [Production and application of 3-phosphoadenosine-5- phosphosulfate]

[4] Christine Kaufmann, et al. J Exp Bot. Sulfated plant peptide hormones

[5] Vitor H Pomin. Eur J Med Chem. Sulfated glycans in inflammation

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Keywords: Inolitazone dihydrochloride, Efatutazone dihydrochloride; CS-7017 dihydrochloride; RS5444 dihydrochloride supplier, PPAR, inhibitors, activators

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