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IHMT-IDH1-053

Cat. No. M42452

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IHMT-IDH1-053 Structure

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Quality Control & Documentation
Biological Activity

IHMT-IDH1-053 is a highly selectivity and irreversible IDH1-mutant inhibitor with an IC50 of 4.7 nM for IDH1 R132H.

Chemical Information
Molecular Weight 532.63
Formula C25H33FN6O4S
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Qianmao Liang et al. Eur J Med Chem. Structure-based discovery of IHMT-IDH1-053 as a potent irreversible IDH1 mutant selective inhibitor

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  Catalog
Abmole Inhibitor Catalog




Keywords: IHMT-IDH1-053 supplier, Isocitrate Dehydrogenase (IDH), inhibitors, activators

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