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ICT5040 is a small molecule CXCR4 antagonist (IC50=3.8 μM). ICT5040 inhibits CXCL12-mediated proliferation and migration, and suppresses CXCL12-induced intracellular calcium mobilisation in U87 glioma cells.
| Molecular Weight | 275.25 |
| Formula | C10H8F3N3OS |
| CAS Number | 215655-21-3 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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