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HTL22562

Cat. No. M21264

All AbMole products are for research use only, cannot be used for human consumption.

HTL22562 Structure

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Quality Control & Documentation
Biological Activity

HTL22562 is a CGRP antagonist intended for use in studies of acute migraine.

Chemical Information
Molecular Weight 763.89
Formula C40H49N11O5
CAS Number 2097085-63-5
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Sarah J Bucknell, et al. J Med Chem. Structure-Based Drug Discovery of N-(( R)-3-(7-Methyl-1 H-indazol-5-yl)-1-oxo-1-((( S)-1-oxo-3-(piperidin-4-yl)-1-(4-(pyridin-4-yl)piperazin-1-yl)propan-2-yl)amino)propan-2-yl)-2'-oxo-1',2'-dihydrospiro[piperidine-4,4'-pyrido[2,3- d][1,3]oxazine]-1-carboxamide (HTL22562): A Calcitonin Gene-Related Peptide Receptor Antagonist for Acute Treatment of Migraine

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Keywords: HTL22562 supplier, CGRP Receptor, inhibitors, activators

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