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HL-8 

Cat. No. M29820

All AbMole products are for research use only, cannot be used for human consumption.

HL-8  Structure

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Quality Control & Documentation
Biological Activity

HL-8 is a PROTAC molecule targeting PI3K kinase. HL-8 has a significant and complete degradation effect on PI3K kinase at a concentration of 10 μM within 8 h. HL-8 has the potential for the research of cancer diseases.

Chemical Information
Molecular Weight 1144.27
Formula C57H59F2N11O9S2
CAS Number 2766352-64-9
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Christopher Wittmann, et al. J Med Chem. Highly Antiproliferative Latonduine and Indolo[2,3- c]quinoline Derivatives: Complex Formation with Copper(II) Markedly Changes the Kinase Inhibitory Profile

[2] Maximilian N Kopylovich, et al. Dalton Trans. Complexes of copper(II) with 3-(ortho-substituted phenylhydrazo)pentane-2,4-diones: syntheses, properties and catalytic activity for cyclohexane oxidation

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  Catalog
Abmole Inhibitor Catalog




Keywords: HL-8  supplier, PI3K, inhibitors, activators

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