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Histrelin acetate

Cat. No. M10505

All AbMole products are for research use only, cannot be used for human consumption.

Histrelin acetate Structure
Size Price Availability Quantity
1mg USD 90 In stock
5mg USD 170 In stock
10mg USD 290 In stock
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Biological Activity

Histrelin is a nonapeptide analog of GnRH (gonadotropin-releasing hormone) with added potency. When present in the bloodstream, it can act on gonadotropes. Histrelin can stimulate these cells to release luteinizing hormone and follicle-stimulating hormone. Histrelin is considered a GnRH agonist. Histrelin acetate is used as a subcutaneous hydrogel implant for the treatment of prostate cancer and for the suppression of gonadal sex hormone production in children with central precocious puberty.

Chemical Information
Molecular Weight 1383.58
Formula C66H86N18O12.XC2H4O2
CAS Number 220810-26-4
Solubility (25°C) Water
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Katherine A Lewis, et al. J Pediatr. A single histrelin implant is effective for 2 years for treatment of central precocious puberty

[2] David Gillis, et al. J Pediatr. Time to menarche and final height after histrelin implant treatment for central precocious puberty

[3] Katherine A Lewis, et al. J Pediatr. Random luteinizing hormone often remains pubertal in children treated with the histrelin implant for central precocious puberty

[4] Neal Shore, et al. BJU Int. Long-term efficacy and tolerability of once-yearly histrelin acetate subcutaneous implant in pаt ιепts with advanced prostate cancer

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Keywords: Histrelin acetate supplier, LHRH/GnRH, inhibitors, activators

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