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Olverembatinib (GZD824) dimesylate is a third-generation oral effective BCR-ABL inhibitor, acting on BCR-ABL (WT) and BCR-ABL (T315I) with IC50 of 0.34 nM and 0.68 nM, respectively.
| Molecular Weight | 724.77 |
| Formula | C29H27F3N6O.2CH4O3S |
| CAS Number | 1421783-64-3 |
| Solubility (25°C) | DMSO 90 mg/mL Water 40 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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| Bosutinib
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| Dasatinib
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| DCC-2036
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