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GSK737

Cat. No. M41652

All AbMole products are for research use only, cannot be used for human consumption.

GSK737 Structure

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Quality Control & Documentation
Biological Activity

GSK737 is a BRD4 BD1 and BD2 inhibitor, with pIC50 values of 5.3 and 7.3 respectively.

Chemical Information
Molecular Weight 363.41
Formula C20H21N5O2
CAS Number 2748687-95-6
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Helen E Aylott et al. J Med Chem. Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors

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  Catalog
Abmole Inhibitor Catalog




Keywords: GSK737 supplier, Epigenetic Reader Domain, inhibitors, activators

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