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GSK256066 Trifluoroacetate

Cat. No. M14503

All AbMole products are for research use only, cannot be used for human consumption.

GSK256066 Trifluoroacetate Structure

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Quality Control & Documentation
Biological Activity

GSK256066 Trifluoroacetate is a selective and high-affinity phosphodiesterase 4 (PDE) inhibitor, with an IC50 of 3.2 pM for PDE4B. GSK256066 Trifluoroacetate is developed for the research of chronic obstructive pulmonary disease.

Chemical Information
Molecular Weight 632.61
CAS Number 1415560-64-3
Solubility (25°C) DMSO 50 mg/mL
Storage 2-8°C, dry, sealed
References

[1] Taruna Joshi, et al. J Pharmacol Exp Ther. GS-5759, a Bifunctional β2-Adrenoceptor Agonist and Phosphodiesterase 4 Inhibitor for Chronic Obstructive Pulmonary Disease with a Unique Mode of Action: Effects on Gene Expression in Human Airway Epithelial Cells

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  Catalog
Abmole Inhibitor Catalog




Keywords: GSK256066 Trifluoroacetate supplier, PDE, inhibitors, activators

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