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GSK 4716

Cat. No. M6165

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GSK 4716 Structure
Size Price Availability Quantity
5mg USD 50 In stock
10mg USD 75 In stock
50mg USD 320 In stock
100mg USD 565 In stock
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Quality Control & Documentation
Biological Activity

GSK 4716 is a selective agonist with estrogen-related receptors ERRβ and ERRγ.

Chemical Information
Molecular Weight 282.33
Formula C17H18N2O2
CAS Number 101574-65-6
Solubility (25°C) 10 mM in DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Saili KS, et al. Toxicology. Neurodevelopmental low-dose bisphenol A exposure leads to early life-stage hyperactivity and learning deficits in adult zebrafish.

[2] Kim Y, et al. J Comb Chem. Efficient discovery of selective small molecule agonists of estrogen-related receptor gamma using combinatorial approach.

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Keywords: GSK 4716 supplier, Estrogen Receptor, inhibitors, activators

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