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GNE-987 is a PROTAC connected by ligands for von Hippel-Lindau and BRD4.
| Molecular Weight | 1096.31 |
| Formula | C56H67F2N9O8S2 |
| CAS Number | 2417371-71-0 |
| Form | Solid |
| Solubility (25°C) | DMSO 100 mg/mL |
| Storage | 4°C, sealed |
| Related PROTAC Products |
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Indisulam is a carbonic anhydrase inibitor and antitumor CDK inhibitor. Indisulam targets the G1 phase of the cell cycle by depleting cyclin E. inducing p53 and p21, and inhibiting CDK2, causing a blockade in the G1/S transition. |
| dBET6
dBET6 is a highly potent, selective and cell-permeable PROTAC connected by ligands for Cereblon and BET, with an IC50 of 14 nM, and has antitumor activity. |
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| MZ 1
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