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GNE-502 

Cat. No. M29052

All AbMole products are for research use only, cannot be used for human consumption.

GNE-502  Structure

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Quality Control & Documentation
Biological Activity

GNE-502 is an orally active and potent degrader for estrogen receptor (ER). GNE-502 can be used for the research of breast cancer.

Chemical Information
Molecular Weight 471.59
Formula C25H30FN3O3S
CAS Number 1953134-16-1
Form Solid
Solubility (25°C) DMSO 100 mg/mL (ultrasonic)
Storage 4°C, protect from light
References

[1] Jason R Zbieg, et al. Bioorg Med Chem Lett. Discovery of GNE-502 as an orally bioavailable and potent degrader for estrogen receptor positive breast cancer

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  Catalog
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Keywords: GNE-502  supplier, Estrogen Receptor, inhibitors, activators

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