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Glesatinib

Cat. No. M30936

All AbMole products are for research use only, cannot be used for human consumption.

Glesatinib Structure
Synonym:

MGCD265

Price and Availability

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Quality Control & Documentation
Biological Activity

Glesatinib (MGCD265) is an orally active, potent MET/SMO dual inhibitor. Glesatinib, a tyrosine kinase inhibitor, antagonizes P-glycoprotein (P-gp) mediated multidrug resistance (MDR) in non-small cell lung cancer (NSCLC).

Chemical Information
Molecular Weight 619.7
Formula C31H27F2N5O3S2
CAS Number 936694-12-1
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Qingbin Cui, et al. Front Oncol. Glesatinib, a c-MET/SMO Dual Inhibitor, Antagonizes P-glycoprotein Mediated Multidrug Resistance in Cancer Cells

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  Catalog
Abmole Inhibitor Catalog




Keywords: Glesatinib, MGCD265 supplier, TAM Receptor, inhibitors, activators

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