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Gemfibrozil

Cat. No. M7822

All AbMole products are for research use only, cannot be used for human consumption.

Gemfibrozil Structure
Synonym:

吉非罗齐; CI-719

Size Price Availability Quantity
100mg USD 55 In stock
500mg USD 105 In stock
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Quality Control & Documentation
Biological Activity

Gemzil is a PPAR-α activator, which is a lipid-lowering agent. Gemfibrozil is also a nonselective inhibitor of P450, with Ki values of 5.8, 24,69 and 82 μM for CYP2C9, 2C19, 2C8 and 1A2, respectively.

Chemical Information
Molecular Weight 250.33
Formula C15H22O3
CAS Number 25812-30-0
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Aleksi Tornio, et al. Role of gemfibrozil as an inhibitor of CYP2C8 and membrane transporters

[2] Barbara S Wiggins, et al. Gemfibrozil in Combination with Statins-Is It Really Contraindicated?

[3] No authors listed. IARC Monogr Eval Carcinog Risks Hum. Gemfibrozil

[4] G J Magarian, et al. Gemfibrozil-induced myopathy

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  Catalog
Abmole Inhibitor Catalog




Keywords: Gemfibrozil, 吉非罗齐; CI-719 supplier, PPAR, inhibitors, activators

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