Free shipping on all orders over $ 500

Fenspiride

Cat. No. M30200

All AbMole products are for research use only, cannot be used for human consumption.

Fenspiride Structure

Price and Availability

For this product's availability, delivery time and price, please email inquiry@abmole.com directly or click the "Inquiry Now" button below.


Quality Control & Documentation
Biological Activity

Fenspiride, an orally active non-steroidal antiinflammatory agent, is an antagonist of H1-histamine receptor. Fenspiride inhibites phosphodiesterase 3 (PDE3), phosphodiesterase 4 (PDE4) and phosphodiesterase 5 (PDE5) activities with -log IC50 values of 3.44, 4.16 and approximately 3.8, respectively. Fenspiride can be used for the research of respiratory diseases.

Chemical Information
Molecular Weight 260.33
Formula C15H20N2O2
CAS Number 5053-06-5
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] R A Kalekin, et al. Sud Med Ekspert. [The study of fenspiride: goals and objectives for chemical and toxicological studies]

[2] Nataliya A Kuzubova, et al. J Smooth Muscle Res. Effect of fenspiride on bronchial smooth muscle of rats with chronic obstructive pulmonary disease

[3] J C Féray, et al. Biochem Pharmacol. Fenspiride and membrane transduction signals in rat alveolar macrophages

[4] C M De Castro, et al. Eur J Pharmacol. Fenspiride: an anti-inflammatory drug with potential benefits in the treatment of endotoxemia

[5] D Bee, et al. Clin Sci (Lond). Effect of fenspiride on pulmonary function in the rat and guinea pig

Related Histamine Receptor Products
Ciproxifan maleate

Ciproxifan is an orally bioavailable, extremely potent histamine H3 inverse agonist/antagonist.

Antazoline hydrochloride

Antazoline hydrochloride is a first generation antihistamine, binding to the histamine H1 receptor and blocking the action of endogenous histamine.

Azacyclonol

Azacyclonol, also known as γ-pipradol, which diminishes hallucinations in psychotic individuals.

Azatadine dimaleate

Azatadine dimaleate is an antihistamine and anticholinergic compound with IC50 of 6.5nM and 10nM, respectively.

Bepotastine Besilate

Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.

  Catalog
Abmole Inhibitor Catalog




Keywords: Fenspiride supplier, Histamine Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2026 AbMole BioScience. All Rights Reserved.