Free shipping on all orders over $ 500

ERB 041

Cat. No. M6717

All AbMole products are for research use only, cannot be used for human consumption.

ERB 041 Structure
Synonym:

ERB-041; Prinaberel

Size Price Availability Quantity
5mg USD 104 In stock
10mg USD 162 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

ERB 041 is a potent and selective estrogen receptor β (ERβ) agonist, with IC50s of 5.4, 3.1, and 3.7 nM for ERβ in humans, rats, and mice, respectively.ERB 041 is more than 200 times more selective for ERβ than for ERα. In addition, ERB 041 inhibits the WNT/β-catenin signaling pathway and induces apoptosis in ovarian cancer cells.

Chemical Information
Molecular Weight 271.24
Formula C15H10FNO3
CAS Number 524684-52-4
Solubility (25°C) DMSO 27.12 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Friedmann, et al. Mol Pharmacol. JX401, a p38α inhibitor containing a 4-benzylpiperidine motif, identified via a novel screening system in yeast.

Related Estrogen Receptor Products
Fulvestrant

Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect.

LY500307

LY500307 is a potent, selective estrogen receptor beta agonist with an EC50 of 0.66 nM.

Calcitriol

Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor. *The compound is unstable in solutions, freshly prepared is recommended

Tamoxifen Citrate (ICI 46474)

Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding.

20-Hydroxyecdysone

20-Hydroxyecdysone (Ecdysterone, 20E) is a naturally occurring ecdysteroid hormone which controls the ecdysis (moulting) and metamorphosis of arthropods.

  Catalog
Abmole Inhibitor Catalog




Keywords: ERB 041, ERB-041; Prinaberel supplier, Estrogen Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2026 AbMole BioScience. All Rights Reserved.