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ENMD-1068 hydrochloride is a selective protease-activated receptor 2 (PAR2) antagonist. ENMD-1068 hydrochloride reduces hepatic stellate cell activation and collagen expression by inhibiting TGF-β1/Smad signaling. ENMD-1068 hydrochloride also inhibits the proliferation of endometrial cells and induces apoptosis of epithelial cells in the lesion. ENMD-1068 hydrochloride can be used in the research of endometriosis and liver fibrosis.
| Molecular Weight | 319.87 |
| Formula | C15H30ClN3O2 |
| CAS Number | 2703451-51-6 |
| Form | Solid |
| Solubility (25°C) | Water 80 mg/mL DMSO 120 mg/mL |
| Storage | 4°C, sealed |
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All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.
Products are for research use only. Not for human use. We do not sell to patients.
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