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Endoxifen

Cat. No. M22289

All AbMole products are for research use only, cannot be used for human consumption.

Endoxifen Structure
Size Price Availability Quantity
5mg USD 50 In stock
10mg USD 78 In stock
25mg USD 155 In stock
50mg USD 260 In stock
100mg USD 420 In stock
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Quality Control & Documentation
Biological Activity

Endoxifen is the key active metabolite of Tamoxifen and an estrogen receptor (ER) modulator with high affinity and specificity for the estrogen receptor and inhibits aromatase activity.Endoxifen has been used in studies related to breast cancer, sclerofibroblastoma, and bipolar disorder.

Chemical Information
Molecular Weight 373.49
Formula C25H27NO2
CAS Number 110025-28-0
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Magnus Bcklund, et al. Oncologist. Topical Endoxifen for Mammographic Density Reduction-A Randomized Controlled Trial

[2] Swaathi Jayaraman, et al. Endocrinology. Endoxifen, an Estrogen Receptor Targeted Therapy: From Bench to Bedside

[3] A B Sanchez-Spitman, et al. Expert Rev Clin Pharmacol. Clinical pharmacokinetics and pharmacogenetics of tamoxifen and endoxifen

[4] V Craig Jordan. J Clin Oncol. Endoxifen: The End, or Are We at the Beginning?

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Keywords: Endoxifen supplier, Estrogen Receptor, inhibitors, activators

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