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EMD 495235

Cat. No. M42397

All AbMole products are for research use only, cannot be used for human consumption.

EMD 495235 Structure

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Quality Control & Documentation
Biological Activity

EMD 495235 is a potent and orally active coagulation factor Xa inhibitor with an IC50 of 5.5 nM and a Ki of 6.8 nM.

Chemical Information
Molecular Weight 451.92
Formula C20H22ClN3O5S
CAS Number 811811-33-3
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Werner W K R Mederski et al. Bioorg Med Chem Lett. Chlorothiophenecarboxamides as P1 surrogates of inhibitors of blood coagulation factor Xa

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Betrixaban

Betrixaban is a highly potent, selective, and orally efficacious factor Xa inhibitor with IC50 of 1.2 nM(inhibition of Factor 10a).

Edoxaban Tosylate Monohydrate

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BMS-740808

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  Catalog
Abmole Inhibitor Catalog




Keywords: EMD 495235 supplier, Factor Xa, inhibitors, activators

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