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Eltoprazine hyrochloride is a serotonin 5-HT1A/1B receptor agonist that has been shown to reduce L-DOPA-induced dyskinesias in in experimental models of Parkinson′s Disease and in human patients. It has Ki values for 5-HT1A, 5-HT1B and 5-HT1C receptors of 40 nM and 52 nM, respectively.
| Molecular Weight | 256.73 |
| Formula | C12H16N2O2 · HCl |
| CAS Number | 98206-09-8 |
| Form | Solid |
| Solubility (25°C) | Water: 10 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[4] Sharon B Wigal, et al. Pharmacokinetic evaluation of eltoprazine
[5] B Olivier, et al. Behavioural pharmacology of the serenic, eltoprazine
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