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Elacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.
| Molecular Weight | 458.63 |
| CAS Number | 722533-56-4 |
| Solubility (25°C) | DMSO 100 mg/mL |
| Storage | 2-8°C, protect from light, dry, sealed |
[1] Katherine G Sanchez, et al. Elacestrant and the Promise of Oral SERDs
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