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DZD1516

Cat. No. M40621

All AbMole products are for research use only, cannot be used for human consumption.

DZD1516 Structure

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Quality Control & Documentation
Biological Activity

DZD1516 is an orally active, potent, reversible, and selective HER2 small molecule tyrosine kinase inhibitors (TKIs) with an IC50 value of 0.56 nM, which completely penetrates the blood-brain barrier. It can be used in studies related to HER2-positive breast cancer.

Chemical Information
Molecular Weight 547.56
Formula C28H27F2N7O3
CAS Number 2387570-00-3
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
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  Catalog
Abmole Inhibitor Catalog




Keywords: DZD1516 supplier, EGFR/HER2, inhibitors, activators

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