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DS08210767 

Cat. No. M29567

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DS08210767  Structure

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Quality Control & Documentation
Biological Activity

DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM.

Chemical Information
Molecular Weight 513.67
Formula C31H39N5O2
CAS Number 2376334-75-5
Form Solid
Solubility (25°C) DMSO 5 mg/mL (ultrasonic and warming and heat to 60°C)
Storage Powder -20°C
References

[1] Yoshikazu Arai, et al. Bioorg Med Chem Lett. Discovery of novel PTHR1 antagonists: Design, synthesis, and structure activity relationships

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Keywords: DS08210767  supplier, Thyroid Hormone Receptor, inhibitors, activators

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