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Delcasertib

Cat. No. M10490

All AbMole products are for research use only, cannot be used for human consumption.

Delcasertib Structure
Synonym:

KAI-9803; BMS-875944

Size Price Availability Quantity
5mg USD 460 In stock
10mg USD 660 In stock
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Quality Control & Documentation
Biological Activity

Delcasertib (KAI-9803) is a potent and selective δ-protein kinase C (δPKC) inhibitor, it could ameliorate injury associated with ischemia and reperfusion in animal models of acute myocardial infarction (MI).

Chemical Information
Molecular Weight 2880.28
Formula C120H199N45O34S2
CAS Number 949100-39-4
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] A Michael Lincoff, et al. Eur Heart J. Inhibition of delta-protein kinase C by delcasertib as an adjunct to primary percutaneous coronary intervention for acute anterior ST-segment elevation myocardial infarction: results of the PROTECTION AMI Randomized Controlled Trial

[2] Yoshihiro Miyaji, et al. Drug Metab Dispos. Distribution of KAI-9803, a novel δ-protein kinase C inhibitor, after intravenous administration to rats

[3] Eric Bates, et al. Circulation. Intracoronary KAI-9803 as an adjunct to primary percutaneous coronary intervention for acute ST-segment elevation myocardial infarction

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Keywords: Delcasertib, KAI-9803; BMS-875944 supplier, PKC, inhibitors, activators

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