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dCBP-1 is a potent and selective heterobifunctional degrader of p300/CBP based on Cereblon ligand. dCBP-1 is exceptionally potent at killing multiple myeloma cells and ablates oncogenic enhancer activity driving MYC expression.
| Molecular Weight | 1028.11 |
| Formula | C51H63F2N11O10 |
| CAS Number | 2484739-25-3 |
| Solubility (25°C) | DMSO 30 mg/mL (ultrasonic and warming) |
| Storage | -20°C, protect from light, dry, sealed |
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