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CY 208-243 

Cat. No. M25551

All AbMole products are for research use only, cannot be used for human consumption.

CY 208-243  Structure

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Quality Control & Documentation
Biological Activity

CY 208-243 is a selective dopamine D1 receptor agonist which exhibits antiparkinsonian activity.

Chemical Information
Molecular Weight 274.36
Formula C19H18N2
CAS Number 100999-26-6
Form Solid
Solubility (25°C) DMSO 40 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] C Gagnon, et al. Neurosci Lett. Chronic CY 208-243 treatment of MPTP-monkeys causes regional changes of dopamine and GABAA receptors

[2] R W Foote, et al. Life Sci. CY 208-243: a unique combination of atypical opioid antinociception and D1 dopaminomimetic properties

[3] A Imperato, et al. Eur J Pharmacol. CY 208-243, a novel dopamine D-1 receptor agonist, fails to modify dopamine release in freely moving rats

[4] B Abbott, et al. Pharmacol Biochem Behav. CY 208-243 behaves as a typical D-1 agonist in the reserpine-treated mouse

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Keywords: CY 208-243  supplier, Dopamine Receptor, inhibitors, activators

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