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CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors.
| Molecular Weight | 391.77 |
| Formula | C19H13ClF3N3O |
| CAS Number | 871362-31-1 |
| Solubility (25°C) | DMSO 60 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Vivek Subbiah, et al. Advances in Targeting RET-Dependent Cancers
[3] Haifeng Zhang, et al. CTEP Versus LESS Totally Extraperitoneal Hernioplasty
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