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Cipralisant

Cat. No. M29275

All AbMole products are for research use only, cannot be used for human consumption.

Cipralisant Structure
Synonym:

GT-2331

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Quality Control & Documentation
Biological Activity

Cipralisant (GT-2331) is an orally active, low-toxicity, potent, selective, high affinity histamine H3 receptor full antagonist in vivo, and an agonist in vitro, with a pKi of 9.9 for histamine H3 receptor and a Ki of 0.47 nM for rat histamine H3 receptor. Cipralisant has the potential for attention-deficit hyperactivity disorder research.

Chemical Information
Molecular Weight 216.32
Formula C14H20N2
CAS Number 213027-19-1
Form Solid
Solubility (25°C) DMSO 200 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Kathleen M Krueger, et al. J Pharmacol Exp Ther. G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations

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  Catalog
Abmole Inhibitor Catalog




Keywords: Cipralisant, GT-2331 supplier, Histamine Receptor, inhibitors, activators

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