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CID 2745687 is a specific, reversible and competitive GPR35 antagonist with a Ki of 12.8 nM. CID 2745687 (pIC50=6.27±0.08) fully reverses the agonist action of Cromolyn disodium. CID 2745687 (CID2745687; 1 mg/kg; administrated orally every day for the last 4 weeks) reverses Lodoxamide-mediated anti-fibrotic effects.
| Molecular Weight | 395.43 |
| Formula | C17H19F2N5O2S |
| CAS Number | 264233-05-8 |
| Solubility (25°C) | DMSO 90 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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