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Cerlapirdine

Cat. No. M30923

All AbMole products are for research use only, cannot be used for human consumption.

Cerlapirdine Structure
Synonym:

SAM-531; PF-05212365

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Quality Control & Documentation
Biological Activity

Cerlapirdine (SAM-531, PF-05212365) is a selective and potent full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine has the potential for researching the Alzheimer's disease.

Chemical Information
Molecular Weight 409.5
Formula C22H23N3O3S
CAS Number 925448-93-7
Form Solid
Solubility (25°C) DMSO 41.67 mg/mL (ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C)
Storage 4°C, protect from light
References

[1] Ramakrishna Nirogi, et al. Biomolecules. Progress in Investigational Agents Targeting Serotonin-6 Receptors for the Treatment of Brain Disorders

[2] Susanna Tse, et al. Drug Metab Dispos. Disposition and metabolic profiling of [(14)C]cerlapirdine using accelerator mass spectrometry

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  Catalog
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Keywords: Cerlapirdine, SAM-531; PF-05212365 supplier, 5-HT Receptor, inhibitors, activators

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