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CCT369260

Cat. No. M21157

All AbMole products are for research use only, cannot be used for human consumption.

CCT369260  Structure

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Quality Control & Documentation
Biological Activity

CCT369260 is an orally active, B-cell lymphoma 6 (BCL6) inhibitor with antitumor activity and an IC50 value of 520 nM.

Chemical Information
Molecular Weight 508.99
Formula C24H31ClF2N6O2
CAS Number 2253878-44-1
Solubility (25°C) DMSO ≥ 200 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Rosemary Huckvale, et al. J Med Chem. Improved Binding Affinity and Pharmacokinetics Enable Sustained Degradation of BCL6 In Vivo

[2] Benjamin R Bellenie, et al. J Med Chem. Achieving In Vivo Target Depletion through the Discovery and Optimization of Benzimidazolone BCL6 Degraders

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  Catalog
Abmole Inhibitor Catalog




Keywords: CCT369260 supplier, Bcl-2, inhibitors, activators

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