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BI 639667

Cat. No. M28125

All AbMole products are for research use only, cannot be used for human consumption.

BI 639667 Structure
Synonym:

CCR1 antagonist 8

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Quality Control & Documentation
Biological Activity

BI 639667 (compound 19n), a third azaindazole series compound, is a CCR1 antagonist, with an IC50 of 1.8 nM in Ca2+ flux assay.

Chemical Information
Molecular Weight 451.47
Formula C22H18FN5O3S
CAS Number 1295298-26-8
Form Solid
Solubility (25°C) DMSO 10 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Scott V Jermain, et al. Mol Pharm. In Vitro and In Vivo Behaviors of KinetiSol and Spray-Dried Amorphous Solid Dispersions of a Weakly Basic Drug and Ionic Polymer†

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  Catalog
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Keywords: BI 639667, CCR1 antagonist 8 supplier, CCR, inhibitors, activators

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