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Camlipixant (BLU-5937) a potent, selective, non-competitive and orally active P2X3 homotrimeric receptor antagonist with an IC50 of 25 nM against hP2X3 homotrimeric.
Camlipixant (500 nM) blocks ATP-mediated dorsal root ganglion (DRG) neuron sensitization.
In vivo, Camlipixant (3-30 mg/kg; oral) reduces histamine- and ATP- induced cough hypersensitivity in guinea pigs. Camlipixant can be used for the research of refractory chronic cough.
| Molecular Weight | 458.46 |
| Formula | C23H24F2N4O4 |
| CAS Number | 1621164-74-6 |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related P2 Receptor Products |
|---|
| Prasugrel hydrochloride
Prasugrel hydrochloride is a novel inhibitor of platelet activation and aggregation. |
| GW 791343 dihydrochloride
GW 791343 dihydrochloride is a non-competitive inhibitor of human P2X(7) receptor. |
| Prasugrel
Prasugrel is a platelet inhibitor irreversibly binding to P2Y12 receptors. |
| MRS 2578
MRS2578 is a potent P2Y6 receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors. |
| PPADS Tetrasodium
PPADS tetrasodium salt is a non-selective P2 purinergic antagonist blocking recombinant P2X1, P2X2, P2X3, P2X5 with IC50 of 1-2.6 μM, native P2Y2-like with IC50 of ~ 0.9 mM, and recombinant P2Y4 receptors with IC50 of ~ 15 mM |
All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.
Products are for research use only. Not for human use. We do not sell to patients.
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