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BRL 54443 is a 5-HT1E and 5-HT1F receptor agonist with pKi of 8.7 and 9.25, respectively, witha weak binding affinity for 5-HT1A, 5-HT1B, 5-HT1D receptors.
| Molecular Weight | 230.31 |
| Formula | C14H18N2O |
| CAS Number | 57477-39-1 |
| Solubility (25°C) | DMSO 30 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Peiyu Xu, et al. Structural insights into the lipid and ligand regulation of serotonin receptors
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