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BMS-986172

Cat. No. M43804

All AbMole products are for research use only, cannot be used for human consumption.

BMS-986172 Structure

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Quality Control & Documentation
Biological Activity

BMS-986172 is an orally active MGAT2 inhibitor with an IC50 of 4.6 nM and 20 nM for hMGAT2 and mMGAT2, respectively. BMS-986172 can be used for the research related to obesity.

Chemical Information
Molecular Weight 589.47
Formula C24H22F7N7O3
CAS Number 1808258-99-2
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Wei Meng et al. J Med Chem. Discovery of 12 (BMS-986172) as a Highly Potent MGAT2 Inhibitor that Achieved Targeted Efficacious Exposures at a Low Human Dose for the Treatment of Metabolic Disorders

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Keywords: BMS-986172 supplier, Transferase, inhibitors, activators

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