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Bms-687453 is an effective and selective PPARα agonist with EC50 and IC50 of 10 nM and 260 nM for human PPARα, respectively. The EC50 and IC50 values were 4100 nM and >15000 nM, respectively.
| Molecular Weight | 444.86 |
| Formula | C22H21ClN2O6 |
| CAS Number | 1000998-59-3 |
| Form | Solid |
| Solubility (25°C) | DMSO > 31 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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