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BI-1347

Cat. No. M13597

All AbMole products are for research use only, cannot be used for human consumption.

BI-1347 Structure
Size Price Availability Quantity
1mg USD 50 In stock
5mg USD 95 In stock
10mg USD 150 In stock
25mg USD 300 In stock
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Quality Control & Documentation
Biological Activity

BI-1347 is a potent CDK8 inhibitor extracted from patent WO2017202719A1, product I-003, has an IC50 of 1.1 nM.

Chemical Information
Molecular Weight 356.42
CAS Number 2163056-91-3
Solubility (25°C) DMSO 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Marco H Hofmann, et al. Mol Cancer Ther. Selective and Potent CDK8/19 Inhibitors Enhance NK-Cell Activity and Promote Tumor Surveillance

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  Catalog
Abmole Inhibitor Catalog




Keywords: BI-1347 supplier, CDK, inhibitors, activators

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