All AbMole products are for research use only, cannot be used for human consumption.
Azelastine hydrochloride (Astelin) is a potent, second-generation, selective, histamine antagonist. Azelastine hydrochloride (Astelin) has a triple mode of action: Anti-histamine effect, mast-cell stabilizing effect and anti-inflammatory effect. Azelastine hydrochloride (Astelin) has a rapid onset of action: 15 minutes with the nasal spray and 3 minutes with the eye drops. The effect lasts for 12 hours.
| Molecular Weight | 418.36 |
| Formula | C22H24ClN3O.HCl |
| CAS Number | 79307-93-0 |
| Solubility (25°C) | DMSO 80 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related Histamine Receptor Products |
|---|
| Ciproxifan maleate
Ciproxifan is an orally bioavailable, extremely potent histamine H3 inverse agonist/antagonist. |
| Antazoline hydrochloride
Antazoline hydrochloride is a first generation antihistamine, binding to the histamine H1 receptor and blocking the action of endogenous histamine. |
| Azacyclonol
Azacyclonol, also known as γ-pipradol, which diminishes hallucinations in psychotic individuals. |
| Azatadine dimaleate
Azatadine dimaleate is an antihistamine and anticholinergic compound with IC50 of 6.5nM and 10nM, respectively. |
| Bepotastine Besilate
Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7. |
All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2026 AbMole BioScience. All Rights Reserved.
