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AZD8154

Cat. No. M21171

All AbMole products are for research use only, cannot be used for human consumption.

AZD8154  Structure

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Quality Control & Documentation
Biological Activity

AZD8154 is a novel inhaled selective PI3Kγδ dual inhibitor targeting airway inflammatory diseases.

Chemical Information
Molecular Weight 551.68
Formula C27H29N5O4S2
CAS Number 2215022-45-8
Solubility (25°C) DMSO : 25 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Gail M Gauvreau, et al. Eur Respir J. Allergen provocation tests in respiratory research: building on 50 years of experience

[2] Muhammad Waqas Sadiq, et al. Br J Clin Pharmacol. Characterisation of pharmacokinetics, safety and tolerability in a first-in-human study for AZD8154, a novel inhaled selective PI3Kγδ dual inhibitor targeting airway inflammatory disease

[3] Matthew W D Perry, et al. J Med Chem. Discovery of AZD8154, a Dual PI3Kγδ Inhibitor for the Treatment of Asthma

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  Catalog
Abmole Inhibitor Catalog




Keywords: AZD8154 supplier, PI3K, inhibitors, activators

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