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AZD 1283 is a high affinity P2Y12 antagonist (Kd = 11 nM). Causes a dose-dependent increase in blood flow and inhibits ADP-induced platelet aggregation in vivo. Antithrombotic.
| Molecular Weight | 470.54 |
| Formula | C23H26N4O5S |
| CAS Number | 919351-41-0 |
| Form | Solid |
| Solubility (25°C) | DMSO 47.05 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Naya, et al. J Med Chem. Design, synthesis, and discovery of a novel CCR1 antagonist.
| Related P2 Receptor Products |
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| Prasugrel
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| MRS 2578
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| PPADS Tetrasodium
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