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Azasetron dihydrochloride

Cat. No. M3201

All AbMole products are for research use only, cannot be used for human consumption.

Azasetron dihydrochloride Structure
Synonym:

Y-25130 2HCl; SENS-401 dihydrochloride

Size Price Availability Quantity
5mg USD 40 In stock
10mg USD 65 In stock
50mg USD 225 In stock
100mg USD 385 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Azasetron dihydrochloride is the hydrochloride form of Azasetron and is also an orally active 5-HT3 receptor antagonist for studies related to ear disorders such as sudden hearing loss.

Chemical Information
Molecular Weight 386.27
Formula C17H20ClN3O3.HCl
CAS Number 123040-16-4
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Bao-Xia Fang, et al. Stability of azasetron-dexamethasone mixture for chemotherapy-induced nausea and vomiting administration

[2] Guanyang Lin, et al. Determination of azasetron hydrochloride in rabbit plasma by liquid chromatography tandem mass spectrometry and its application

[3] Yasuhiko Yamada, et al. Analysis of antiemetic effect of various dosage regimens of azasetron hydrochloride based on 5-HT3 receptor occupancy of serotonin

[4] K Katayama, et al. High affinity binding of azasetron hydrochloride to 5-hydroxytryptamine3 receptors in the small intestine of rats

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Keywords: Azasetron dihydrochloride, Y-25130 2HCl; SENS-401 dihydrochloride supplier, 5-HT Receptor, inhibitors, activators

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