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AZ13824374

Cat. No. M21069

All AbMole products are for research use only, cannot be used for human consumption.

AZ13824374  Structure

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Quality Control & Documentation
Biological Activity

AZ13824374 is an in vitro ATAD2 inhibitor with anti-proliferative activity against breast cancer. pIC50 of AZ13824374 against ATAD2 in the ATAD2 FRET and ATAD2 NanoBRET assays were 8.2 and 6.2, respectively.

Chemical Information
Molecular Weight 562.68
Formula C30H39FN8O2
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jiahui Fu, et al. Theranostics. ATPase family AAA domain-containing protein 2 (ATAD2): From an epigenetic modulator to cancer therapeutic target

[2] Jon J Winter-Holt, et al. J Med Chem. Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models

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  Catalog
Abmole Inhibitor Catalog




Keywords: AZ13824374 supplier, Epigenetic Reader Domain, inhibitors, activators

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