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AS2521780 

Cat. No. M27957

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AS2521780  Structure

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Quality Control & Documentation
Biological Activity

AS2521780 is a novel PKCθ selective inhibitor with an IC50 of 0.48 nM.

Chemical Information
Molecular Weight 547.76
Formula C30H41N7OS
CAS Number 1214726-89-2
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Hidehiko Fukahori, et al. Int Immunopharmacol. Effect of novel PKCθ selective inhibitor AS2521780 on acute rejection in rat and non-human primate models of transplantation

[2] Hidehiko Fukahori, et al. Eur J Pharmacol. Effect of AS2521780, a novel PKCθ selective inhibitor, on T cell-mediated immunity

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  Catalog
Abmole Inhibitor Catalog




Keywords: AS2521780  supplier, PKC, inhibitors, activators

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