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AR-C 118925XX

Cat. No. M6457

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AR-C 118925XX Structure
Synonym:

ARC118925XX

Size Price Availability Quantity
1mg USD 185 In stock
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Quality Control & Documentation
Biological Activity

AR-C 118925XX is a selective, competitive P2Y2 receptor antagonist. AR-C 118925XX is inactive against a panel of 37 other receptors at a concentration of 10 μM. AR-C 118925XX inhibits ATP-γS-induced mucin secretion in bronchial epithelial cells (IC50 = 1 μM). AR-C 118925XX inhibits P2Y2 receptor-induced β-arrestin translocation in vitro (pA2 = 37.2-51.3 nM).

Chemical Information
Molecular Weight 537.59
Formula C28H23N7O3S
CAS Number 216657-60-2
Solubility (25°C) DMSO 53.76 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Aloyo and Harvey. Eur J Pharmacol. Antagonist binding at 5-HT2A and 5-HT2C receptors in the rabbit: high correlation with the profile for the human receptors.

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Keywords: AR-C 118925XX, ARC118925XX supplier, P2 Receptor, inhibitors, activators

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