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AR-A 2 is a selective 5-HT1B receptor antagonist, with high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki=0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki, 5 nM), and shows an EC50 of 4.5 nM for the guinea pig 5-HT1B receptor; AR-A 2 can be used in the research of depression and anxiety.
| Molecular Weight | 448.6 |
| Formula | C27H36N4O2 |
| CAS Number | 220051-79-6 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
[2] Yuan Zhang, et al. Allergy. Advances and highlights in allergic rhinitis
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